Pharmokinetics of Premedication Drugs

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58 Questions

Which receptor is primarily associated with analgesic and sedation effects in the brain?

Mu receptors

Which drug is more selective for the alpha 2 medication compared to Xylazine and Medetomidine?

Dexmedetomidine

Which opioid is a partial agonist and will not elicit a fuller response even at maximal dose?

Buprenorphine

Which drug can act as a reverser for A2 adrenoreceptor agonists?

Atipamezole

Which receptor is associated with marked bradycardia and hypertension?

Alpha 2 receptor

Which class of drugs primarily acts by antagonizing dopamine receptors?

Phenothiazines

Which receptor is primarily associated with analgesic and anti-depressant effects in the brain?

Delta receptors

Which receptor is primarily associated with analgesic, sedative, and diuretic effects in the brain?

Kappa receptors

Which receptor is primarily associated with analgesia, sedation, respiratory depression, euphoria, and constipation in the brain?

Mu receptors

Which receptor is primarily associated with anxiety and depression in the brain, spinal cord, and amygdala?

Nociception receptors

Which of the following characteristics is important for a drug used for premedication?

Rapid onset

What is the role of lipophilicity in premedication drugs?

To cross plasma membranes

Which of the following is a characteristic of centrally acting drugs?

Inhibitory effects

What is the role of alpha 2 adrenoreceptor agonists?

Constriction or relaxation

What is the main reason for using selective alpha 2 drugs?

To bind to A2 receptors only

Which of the following is a property of alpha 2 adrenoreceptor agonists?

Sedative and muscle relaxant properties

Which of the following is should not be a characteristic of a premedication drugs?

Long elimination time

What is the role of A2 receptors in the cholinergic system?

Reduction of noradrenaline release

What is the effect of increasing the dose of alpha 2 adrenoreceptor agonists?

Increased chance of affecting other receptors

Which of the following drugs is a selective alpha 2 adrenoreceptor agonist?

Medetomidine

Which opioid is commonly used in veterinary medicine as an analgesic?

Butorphanol

Which receptor is primarily associated with analgesia, sedation, respiratory depression, euphoria, and constipation in the brain?

Mu receptor

Which of the following is a characteristic of benzodiazepines?

Causes anxiolysis, sedation, and hypnosis

Which drug is a NMDA receptor antagonist?

Ketamine

Which of the following is a property of ketamine?

Rapid onset of action and short duration

Which receptor is primarily associated with analgesic and anti-depressant effects in the brain?

Delta receptor

Which of the following is a property of phenothiazines?

Antagonism of dopamine receptors

Which receptor is primarily associated with analgesic, sedative, and diuretic effects in the brain?

Kappa receptor

Which of the following characteristics is important for a drug used for premedication?

Must be lipophilic

What is the role of lipophilicity in premedication drugs?

It allows the drug to distribute to the brain

What is the effect of increasing the dose of alpha 2 adrenoreceptor agonists?

Increase the chance to effect other receptors

Which receptor is primarily associated with analgesic, sedative, and muscle relaxant properties in the brain?

Alpha 2 adrenoreceptor

Which receptor is primarily associated with heart function, airways, and metabolic effects?

Beta adrenoreceptor

Which of the following is a property of alpha 2 adrenoreceptor agonists?

Marked bradycardia and hypotension

Which drug is more selective for the alpha 2 receptor compared to Xylazine?

Medetomidine

What is the main reason for using selective alpha 2 drugs?

To bypass the blood-brain barrier

What is the role of A2 receptors in the cholinergic system?

Inhibits the release of noradrenaline

Which of the following is NOT associated with alpha 2 adrenoreceptor agonists?

Euphoric effects

Which of the following drugs is a selective alpha 2 adrenoreceptor agonist?

Medetomidine

Which receptor is primarily associated with analgesic, sedative, and diuretic effects in the brain?

Kappa receptors

What is the main reason for using selective alpha 2 drugs?

To provide analgesia

Which receptor is associated with marked bradycardia and hypertension?

Alpha 2 receptors

Which of the following is NOT a characteristic of premedication drugs?

Rapid onset of action

Which opioid is a partial agonist and will not elicit a fuller response even at maximal dose?

Buprenorphine

Which of the following is NOT associated with alpha 2 adrenoreceptor agonists?

Axiolysis

Which drug can act as a reverser for A2 adrenoreceptor agonists?

Atipamezole

What is the role of lipophilicity in premedication drugs?

It aids in oral and intramuscular absorption

Which of the following is a property of benzodiazepines?

They act as GABA agonists

Which characteristic is important for a drug used for premedication?

Must be lipophilic and readily absorbed

Which receptor is primarily associated with analgesic effects in the brain?

Alpha 2 adrenoreceptor

What is the effect of increasing the dose of alpha 2 adrenoreceptor agonists?

Increase the chance to effect other receptors not A2 specific

What is the role of A2 receptors in the cholinergic system?

Promote the action of inhibitory neurotransmitters

Which of the following is a characteristic of benzodiazepines?

Crosses the blood brain barrier

Which receptor is associated with marked bradycardia and hypotension?

Alpha 2 adrenoreceptor

What is the main reason for using selective alpha 2 drugs?

To promote the action of inhibitory neurotransmitters

Which receptor is primarily associated with sedation and muscle relaxation in the brain?

Alpha 2 adrenoreceptor

Which of the following drugs is a selective alpha 2 adrenoreceptor agonist?

Xylazine

Which of the following characteristics is important for a drug used for premedication?

Must be lipophilic and readily absorbed

Test your knowledge on drugs used for premedication and their characteristics with this quiz. Learn why premedication is important and what qualities a drug needs to have for effective premedication. Explore concepts like rapid onset, absorption, lipophilicity, and central action. Challenge yourself and expand your understanding of premedication drugs.

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