Fioricet Drugs Flashcards

Questions and Answers

What is the brand name of butalbital, acetaminophen, & caffeine?

Fioricet

What drug class does butalbital, acetaminophen, & caffeine belong to?

Analgesic

What is the labeled indication of use for butalbital, acetaminophen, & caffeine?

Relief of the symptom complex tension (or muscle contraction) headache

What is the dosage form of butalbital, acetaminophen, & caffeine?

Tablets Signup and view all the answers

What is the MOA for butalbital, acetaminophen, & caffeine? (List 3)

Acetaminophen: Produces analgesia by inhibiting prostaglandin synthesis in the CNS and through a peripheral action of blocking pain impulse generation; Butalbital: Produces sensory cortex depression through inhibition of conduction in the reticular formation at the level of the thalamus; Caffeine: Produces CNS stimulation by inhibition of phosphodiesterase which increases the accumulation of c-AMP Signup and view all the answers

What are the adverse effects of butalbital, acetaminophen, & caffeine? (List 3)

Dizziness, drowsiness, lightheadedness Signup and view all the answers

What is the pregnancy category for butalbital, acetaminophen, & caffeine?

C Signup and view all the answers

What are the other counseling points for butalbital, acetaminophen, & caffeine? (List 7)

<ol> <li>May cause drowsiness. Use caution while operating machinery or when mental alertness is required; 2. Avoid alcohol while taking this medication; 3. May take with food or milk to avoid GI upset; 4. Do not exceed prescribed dosage; 5. WARNING: This medication may be habit-forming; 6. Contact a physician if the above side effects are severe or persistent; 7. If a dose is missed, skip it and return to normal dosing schedule.</li> </ol> Signup and view all the answers

What are the storage instructions for butalbital, acetaminophen, & caffeine?

Store in a cool, dry place away from sunlight and children. Signup and view all the answers

Study Notes

Fioricet Overview

Fioricet is the brand name for butalbital, acetaminophen, and caffeine.
Classified as an analgesic, primarily used for headache relief.

Indications

Labeled for relief of tension or muscle contraction headaches.

Dosage Form

Available in tablet form for administration.

Mechanism of Action (MOA)

Acetaminophen: Analgesic effect achieved by inhibiting prostaglandin synthesis in the central nervous system (CNS) and blocking pain impulse generation peripherally.
Butalbital: Depresses sensory cortex by inhibiting conduction in the reticular formation at the thalamus level.
Caffeine: Acts as a CNS stimulant by inhibiting phosphodiesterase, increasing cAMP accumulation.

Adverse Effects

Common side effects include dizziness, drowsiness, and lightheadedness.

Pregnancy Category

Classified as Category C, indicating risk cannot be ruled out during pregnancy.

Counseling Points

Caution advised due to potential drowsiness; avoid operating heavy machinery or activities requiring mental alertness.
Alcohol intake should be avoided while on this medication.
Can be taken with food or milk to minimize gastrointestinal upset.
Patients should not exceed the prescribed dosage.
Warning regarding potential habit-forming nature of the medication.
Seek medical advice if severe or persistent side effects occur.
If a dose is missed, skip it and resume normal dosing schedule.

Storage Instructions

Store in a cool, dry environment, away from sunlight and out of reach of children.

Description

Test your knowledge about Fioricet, a medication containing butalbital, acetaminophen, and caffeine. This quiz covers its brand name, drug class, and indications for use. Perfect for students in pharmacology or healthcare.